Development and characterization of an aptamer binding ligand of fractalkine using domain targeted SELEX.

نویسندگان

  • Brett Waybrant
  • Timothy R Pearce
  • Ping Wang
  • Srinand Sreevatsan
  • Efrosini Kokkoli
چکیده

Fractalkine (FKN) is a unique cell surface protein with potential as a therapeutic target because of its role in inflammatory diseases and cancer. We developed an aptamer, named FKN-S2, with a dissociation constant of 3.4 ± 0.7 nM that is specific to the chemokine domain of fractalkine.

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عنوان ژورنال:
  • Chemical communications

دوره 48 80  شماره 

صفحات  -

تاریخ انتشار 2012